825:
700:
526:
503:
36:
142:
944:
for women has also been studied. The first report of this method claimed a first year failure rate of 3.1%. However, despite a multitude of clinical studies on the use of mepacrine and female sterilization, no randomized, controlled trials have been reported to date and there is some controversy
974:
In the United States, this method has undergone Phase I clinical testing. The FDA has waived the necessity for Phase II clinical trials because of the extensive data pertaining to other uses of mepacrine. The next step in the FDA approval process in the United States is a Phase III large
1373:
Haïk S, Brandel J, Salomon D, Sazdovitch V, Delasnerie-Lauprêtre N, Laplanche J, Faucheux B, Soubrié C, Boher E, Belorgey C, Hauw J, Alpérovitch A (28 December 2004). "Compassionate use of quinacrine in
Creutzfeldt–Jakob disease fails to show significant effects".
736:-resistant giardiasis and patients who should not receive or cannot tolerate metronidazole. Giardiasis with a high level of drug resistance may even require a combination of mepacrine and metronidazole to cure.
1746:
1279:
932:
include inefficient penetration of the blood–brain barrier, as well as the existence of drug-resistant prion proteins that increase in number when selected for by treatment with mepacrine.
824:
1417:
Barret A, Tagliavini F, Forloni G, Bate C, Salmona M, Colombo L, De Luigi A, Limido L, Suardi S, Rossi G, Auvré F, Adjou K, Salès N, Williams A, Lasmézas C, Deslys J (August 2003).
959:
insertion. The procedure is undertaken twice, first in the proliferative phase, 6 to 12 days following the first day of the menstrual cycle and again one month later. The
916:. Small trials in Japan have reported improvement in the condition of patients with the disease, although other reports have shown no significant effect, and treatment of
3745:
1137:
Wall JE, Buijs-Wilts M, Arnold JT, et al. (1995). "A flow cytometric assay using mepacrine for study of uptake and release of platelet dense granule contents".
1570:
Zipper J, Cole LP, Goldsmith A, Wheeler R, Rivera M (1980). "Quinacrine hydrochloride pellets: preliminary data on a nonsurgical method of female sterilisation".
5086:
1789:
182:
1231:"Randomized clinical study of five days apostrophe therapy with mebendazole compared to quinacrine in the treatment of symptomatic giardiasis in children"
5016:
779:
visualization of cells, especially platelets. Mepacrine is a green fluorescent dye taken up by most cells. Platelets store mepacrine in dense granules.
2510:
1712:
1655:
1468:"A possible pharmacological explanation for quinacrine failure to treat prion diseases: pharmacokinetic investigations in a ovine model of scrapie"
5185:
4750:
4347:
4342:
2587:
637:
InChI=1S/C23H30ClN3O/c1-5-27(6-2)13-7-8-16(3)25-23-19-11-9-17(24)14-22(19)26-21-12-10-18(28-4)15-20(21)23/h9-12,14-16H,5-8,13H2,1-4H3,(H,25,26)
1669:
Peterson, H.B., Lubell, L., DeStefano, F., and Ory, H.W. (1983). "The safety and efficacy of tubal sterilization: an international overview".
595:
4265:
3738:
164:
4604:
2805:
1866:
609:
1507:
5041:
4609:
3559:
3550:
1782:
986:. Nevertheless, in 1998 the Supreme Court of India banned the import or use of the drug, allegedly based on reports that it could cause
4614:
3555:
3731:
2735:
1098:"The reduction of serum B-lymphocyte activating factor levels following quinacrine add-on therapy in systemic lupus erythematosus"
2998:
1053:
5136:
4574:
3466:
3282:
3133:
1775:
1642:
Background Paper for the World Health
Organization Consultation on the Development of New Technologies for Female Sterilization
1007:
1767:
3689:
2942:
2503:
2454:
1010:
operatives yellowed their skin using mepacrine tablets in order to more closely match the skin color of their
Chinese peers.
1284:
711:
5140:
4885:
3775:
100:
1747:"How naked World War II sailors ended up riding Mongolian ponies in the Gobi Desert to shoot bazookas at the Japanese"
72:
5180:
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654:
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119:
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3428:
2959:
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5210:
3962:
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256:
79:
5165:
5144:
4855:
4676:
3975:
3084:
2976:
2326:
57:
1299:"Lysosomotropic Agents and Cysteine Protease Inhibitors Inhibit Scrapie-Associated Prion Protein Accumulation"
5170:
4996:
4624:
1890:
905:
796:
5175:
5116:
2557:
1727:
866:
in
Germany first synthesised mepacrine in 1931. The product was one of the first synthetic substitutes for
740:
521:
374:
86:
4966:
4504:
3630:
2991:
765:
744:
482:
4685:
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3931:
3754:
443:
53:
17:
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68:
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3869:
2170:
1519:
Ghaemmaghami S, Ahn M, Lessard P, Giles K, Legname G, et al. (November 2009). Mabbott N (ed.).
5205:
3032:
1003:
941:
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3694:
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2459:
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2298:
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776:
707:
154:
46:
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3908:
2984:
2903:
2685:
2309:
2185:
2141:
1857:
1797:
983:
982:
Many peer reviewed studies suggest that mepacrine sterilization (QS) is potentially safer than
688:
464:
225:
775:
In addition to medical applications, mepacrine is an effective in vitro research tool for the
699:
5195:
4689:
3966:
3944:
3495:
2842:
2693:
2689:
2315:
1706:
1649:
1640:
Sokal, D.C., Kessel. E., Zipper. J., and King. T. (1994). "Quinacrine: Clinical experience".
423:
5120:
4431:
4421:
3638:
3522:
2873:
2603:
2235:
383:
235:
1466:
Gayrard V, Picard-Hagen N, Viguié C, Laroute V, Andréoletti O, Toutain P (February 2005).
1083:
205:
8:
4559:
4283:
3671:
3359:
2743:
2724:
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2436:
1802:
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852:
761:
prophylaxis in patients at high risk of recurrence, e.g., in those with cystic fibrosis.
363:
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1668:
525:
502:
298:
5190:
4735:
4716:
4712:
4698:
4694:
4464:
3917:
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3222:
2666:
2548:
2408:
2215:
1997:
1900:
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1492:
1467:
1399:
1387:
1257:
1230:
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748:
747:
and subcutaneous lupus manifestations, particularly in patients who are unable to take
93:
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1298:
4901:
4875:
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4653:
4644:
4205:
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1946:
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4185:
4101:
3760:
3533:
3501:
3023:
2004:
1983:
1678:
1579:
1542:
1532:
1521:"Continuous Quinacrine Treatment Results in the Formation of Drug-Resistant Prions"
1487:
1479:
1438:
1430:
1383:
1318:
1310:
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1201:
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3124:
2953:
2881:
2850:
2779:
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2678:
2637:
2614:
2579:
2465:
2124:
1975:
1806:
909:
840:
by Allied forces fighting in North Africa and the Far East to prevent malaria.
764:
Mepacrine is not the drug of choice because side effects are common, including
732:
Mepacrine is used off label as a primary antimicrobial agent for patients with
1964:
5159:
4961:
4407:
4071:
4051:
4016:
3824:
3432:
3385:
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2210:
2195:
2088:
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2008:
1923:
1096:
Toubi E, Kessel A, Rosner I, Rozenbaum M, Paran D, Shoenfeld Y (2006).
1034:
960:
848:
769:
726:
684:
571:
354:
5082:
5051:
5036:
5012:
4951:
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3807:
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3272:
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2762:
2575:
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2205:
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2013:
1819:
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forming over a six-week interval to close off the tubes permanently.
921:
792:
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691:, as of August 2020 it is totally unavailable in the United States.
35:
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4640:
4544:
4520:
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4411:
4371:
4313:
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3840:
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3661:
3596:
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2919:
2720:
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900:
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470:
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3057:
2607:
2398:
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867:
1465:
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3791:
3147:
1182:"Resistance to chloroquine unhinges vivax malaria therapeutics"
987:
952:
434:
4575:
2288:
1228:
928:
has also shown no effect. Possible reasons for the lack of an
4825:
4649:
4170:
3803:
963:
effects of the drugs at the utero-tubal junctions (where the
925:
895:
863:
585:
414:
141:
1372:
951:
of mepacrine are inserted through the cervix into a woman's
487:
4886:
3776:
1518:
1416:
1346:
Kobayashi Y, Hirata K, Tanaka H, Yamada T (July 2003). "".
1345:
975:
multi-center clinical trial. The method is currently used
968:
394:
1569:
1095:
1054:"Quinacrine Shortage & What the ACR Is Doing about It"
904:, and full clinical trials of its use as a treatment for
808:
710:); this sign was posted at the 363rd Station Hospital on
955:
using a preloaded inserter device, similar in manner to
1419:"Evaluation of Quinacrine Treatment for Prion Diseases"
1229:
Canete R, Escobedo AA, Gonzalez ME, Almirall P (2006).
935:
4856:
898:
protein and prevent the formation of prion aggregates
739:
Mepacrine is also used off-label for the treatment of
679:, is a medication with several uses. It is related to
4997:
4625:
1613:"Quinacrine sterilization: reports on 40,252 cases".
1136:
1572:
International
Journal of Gynecology & Obstetrics
832:
Mepacrine was initially approved in the 1930s as an
4505:
3753:
1615:
International
Journal of Gynaecology and Obstetrics
1296:
791:is uncertain, but it is thought to act against the
60:. Unsourced material may be challenged and removed.
4392:
5157:
322:
4929:
297:
4806:
4580:Tooltip Phenylethanolamine N-methyltransferase
3909:
855:), and has been researched as an inhibitor of
3739:
2992:
2504:
1783:
1079:
1077:
1075:
1073:
1071:
4432:
1711:: CS1 maint: multiple names: authors list (
1654:: CS1 maint: multiple names: authors list (
1512:
889:
4891:Tooltip Acetylserotonin O-methyltransferase
3781:Tooltip Aromatic L-amino acid decarboxylase
1222:
1089:
795:'s cell membrane. It is known to act as a
617:CCN(CC)CCCC(C)Nc1c2ccc(cc2nc3c1cc(cc3)OC)Cl
204:
3918:
3746:
3732:
2999:
2985:
2511:
2497:
1790:
1776:
1297:Doh-Ura K, Iwaki T, Caughey B (May 2000).
1068:
882:In addition it has been used for treating
524:
501:
362:
3890:
1739:
1546:
1536:
1491:
1442:
1322:
1256:
1246:
1205:
1113:
382:
120:Learn how and when to remove this message
1339:
1179:
894:Mepacrine has been shown to bind to the
823:
698:
175:Micromedex Detailed Consumer Information
5067:
1763:National Institute on Aging (NIA) trial
1459:
497:
342:
14:
5158:
4861:Tooltip Serotonin N-acetyl transferase
1728:"Govt drags feet on quinacrine threat"
1725:
1410:
1290:
1008:Sino-American Cooperative Organization
940:The use of mepacrine for non-surgical
847:is also approved for the treatment of
768:, and may cause permanent damage. See
515:
5186:Experimental methods of birth control
5002:Tooltip Histamine N-methyltransferase
4630:Tooltip Catechol-O-methyl transferase
3727:
2980:
2492:
1771:
836:. It was used extensively during the
717:The main uses of mepacrine are as an
463:
442:
422:
173:
1366:
936:Non-surgical sterilization for women
712:Papua New Guinea during World War II
704:These men didn't take their Atabrine
469:
272:′-(6-Chloro-2-methoxy-acridin-9-yl)-
194:
58:adding citations to reliable sources
29:
4510:Tooltip Dopamine beta-monooxygenase
687:. Although formerly available from
402:
313:
24:
1584:10.1002/j.1879-3479.1980.tb00496.x
1388:10.1212/01.wnl.0000148596.15681.4d
1151:10.1111/j.1365-2141.1995.tb03315.x
25:
5222:
4397:Tooltip Phenylalanine hydroxylase
1756:
1726:George, Nirmala (July 25, 1998).
1621:(Suppl 2): S1–159. October 2003.
743:, indicated in the treatment of
3429:Glutamate-gated chloride channel
1435:10.1128/JVI.77.15.8462-8469.2003
1315:10.1128/JVI.74.10.4894-4897.2000
1115:10.1111/j.1365-3083.2006.01737.x
877:
819:
787:Its mechanism of action against
558:
555:
549:
140:
34:
4934:Tooltip Histidine decarboxylase
1719:
1662:
1633:
1606:
1563:
694:
642:Key:GPKJTRJOBQGKQK-UHFFFAOYSA-N
45:needs additional citations for
4811:Tooltip Tryptophan hydroxylase
4591:Norepinephrine (noradrenaline)
4525:Norepinephrine (Noradrenaline)
3950:Norepinephrine (noradrenaline)
3914:Tooltip Aldehyde dehydrogenase
2327:piperaquine/dihydroartemisinin
1273:
1173:
1130:
1046:
564:
543:
13:
1:
5137:Monoamine reuptake inhibitors
5117:Receptor/signaling modulators
1891:trimethoprim/sulfamethoxazole
1086:Retrieved on August 24, 2009.
1040:
967:enter the uterus) results in
870:although later superseded by
4437:Tooltip Tyrosine hydroxylase
2289:Fixed-dose (co-formulated)
1683:10.1016/0020-7292(83)90051-6
1538:10.1371/journal.ppat.1000673
1285:Dorland's Medical Dictionary
1186:Antimicrob. Agents Chemother
828:Atabrine and mosquito poster
803:inhibitor. It also inhibits
782:
741:systemic lupus erythematosus
7:
5097:Pimagedine (aminoguanidine)
4967:Alpha-Fluoromethylhistidine
1013:
997:
280:-diethylpentane-1,4-diamine
10:
5227:
5141:Monoamine releasing agents
3907:Substrates→Products (with
3467:+esafoxolaner/praziquantel
3283:+esafoxolaner/eprinomectin
3134:+esafoxolaner/eprinomectin
814:
533:Chemical and physical data
5109:
5065:
4995:
4927:
4918:
4884:
4854:
4804:
4783:
4623:
4573:
4503:
4430:
4390:
4364:
4255:
4130:
3902:
3895:Tooltip Monoamine oxidase
3888:
3774:
3767:
3684:
3571:
3512:
3427:
3374:
3358:
3264:
3236:
3221:
3110:
3083:
3055:
3040:
3033:Antiplatyhelmintic agents
3031:
2937:
2872:
2841:
2770:
2761:
2734:
2665:
2628:
2556:
2547:
2538:
2449:
2425:
2397:
2371:
2335:
2279:
2224:
2184:
2171:sulfadoxine/pyrimethamine
2163:
2140:
2096:
2087:
2053:
2027:
1974:
1963:
1954:
1945:
1936:
1899:
1881:
1856:
1840:
1829:
1818:
906:Creutzfeldt–Jakob disease
890:Creutzfeldt–Jakob disease
650:
625:
605:
583:
570:
537:
532:
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481:
453:
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252:
247:
234:
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139:
5181:Sterilization (medicine)
4595:Epinephrine (adrenaline)
3928:Epinephrine (adrenaline)
1671:Int. J. Gynaecol. Obstet
1248:10.3748/wjg.v12.i39.6366
1004:Second Sino-Japanese War
5072:Tooltip Diamine oxidase
2686:Pentavalent antimonials
2558:African trypanosomiasis
2322:artesunate/pyronaridine
2299:artemether/lumefantrine
5211:Diethylamino compounds
4972:Histidine methyl ester
2310:artesunate/amodiaquine
1484:10.1038/sj.bjp.0706072
1235:World J. Gastroenterol
1084:Drugs.com: Quinacrine.
984:surgical sterilization
829:
772:for more information.
725:, and an intrapleural
714:
689:compounding pharmacies
671:or by the trade names
5166:Disulfiram-like drugs
5145:Monoamine neurotoxins
5087:Imidazole acetic acid
2694:Sodium stibogluconate
2690:Meglumine antimoniate
2344:artesunate/mefloquine
2316:artesunate/mefloquine
908:are under way in the
827:
702:
5171:Antiprotozoal agents
5080:Substrates→Products:
5010:Substrates→Products:
4942:Substrates→Products:
4899:Substrates→Products:
4869:Substrates→Products:
4819:Substrates→Products:
4638:Substrates→Products:
4588:Substrates→Products:
4518:Substrates→Products:
4445:Substrates→Products:
4422:3,4-Dihydroxystyrene
4405:Substrates→Products:
3789:Substrates→Products:
3639:naphthalenesulfonate
3523:tetrahydropyrimidine
3360:Antinematodal agents
2604:naphthalenesulfonate
2356:quinine/tetracycline
2028:4-Methanolquinolines
1803:antiprotozoal agents
1198:10.1128/aac.01296-10
54:improve this article
5176:Antimalarial agents
4560:Phenopicolinic acid
4284:Desmethylselegiline
3672:Tetrachloroethylene
2353:quinine/doxycycline
2350:quinine/clindamycin
2338:(not co-formulated)
992:ectopic pregnancies
853:intestinal parasite
136:
4736:2-Hydroxyestradiol
4717:4-Methoxyestradiol
4713:4-Hydroxyestradiol
4699:2-Methoxyestradiol
4695:2-Hydroxyestradiol
4465:2-Hydroxyestradiol
3711:Never to phase III
3589:Diethylcarbamazine
2964:Never to phase III
2476:Never to phase III
2336:Other combinations
2216:dihydroartemisinin
1998:hydroxychloroquine
1348:Rinsho Shinkeigaku
830:
801:-methyltransferase
749:hydroxychloroquine
715:
132:
5153:
5152:
5148:
5105:
5104:
5017:N-Methylhistamine
4947:
4914:
4913:
4902:N-Acetylserotonin
4876:N-Acetylserotonin
4846:Telotristat ethyl
4841:Fenclonine (PCPA)
4798:
4779:
4778:
4654:Homovanillic acid
4645:3-Methoxytyramine
4454:
4384:
4360:
4359:
4356:
4355:
4337:
4278:
4206:tetrahydroharmine
4186:Harmala alkaloids
3981:3-Methoxytyramine
3836:
3815:
3794:
3721:
3720:
3680:
3679:
3354:
3353:
3350:
3349:
3217:
3216:
2974:
2973:
2933:
2932:
2757:
2756:
2711:phosphorylcholine
2661:
2660:
2486:
2485:
2421:
2420:
2393:
2392:
2389:
2388:
2367:
2366:
2363:
2362:
2275:
2274:
2180:
2179:
2083:
2082:
1932:
1931:
1858:Cryptosporidiosis
1180:Baird JK (2011).
1102:Scand. J. Immunol
834:antimalarial drug
708:anti-malaria drug
662:
661:
596:Interactive image
483:CompTox Dashboard
159:Atabrine, Atebrin
130:
129:
122:
104:
16:(Redirected from
5218:
5111:
5073:
5069:
5003:
4999:
4945:
4935:
4931:
4925:
4924:
4892:
4888:
4862:
4858:
4812:
4808:
4802:
4801:
4788:
4741:2-Hydroxyestrone
4726:4-Methoxyestrone
4722:4-Hydroxyestrone
4708:2-Methoxyestrone
4704:2-Hydroxyestrone
4631:
4627:
4581:
4577:
4511:
4507:
4470:2-Hydroxyestrone
4455:-DOPA (levodopa)
4452:
4438:
4434:
4398:
4394:
4388:
4387:
4369:
4335:
4276:
4263:MAO-B selective:
4138:MAO-A-selective:
4102:Phenoxypropazine
3924:
3920:
3915:
3911:
3900:
3899:
3896:
3892:
3834:
3813:
3795:-DOPA (levodopa)
3792:
3782:
3778:
3772:
3771:
3748:
3741:
3734:
3725:
3724:
3534:pyrantel pamoate
3502:Milbemycin oxime
3372:
3371:
3366:macrofilaricides
3234:
3233:
3053:
3052:
3047:schistosomicides
3038:
3037:
3001:
2994:
2987:
2978:
2977:
2768:
2767:
2554:
2553:
2545:
2544:
2513:
2506:
2499:
2490:
2489:
2286:
2285:
2094:
2093:
1972:
1971:
1961:
1960:
1952:
1951:
1943:
1942:
1854:
1853:
1838:
1837:
1827:
1826:
1809:antiparasitics (
1792:
1785:
1778:
1769:
1768:
1751:
1750:
1743:
1737:
1735:
1723:
1717:
1716:
1710:
1702:
1666:
1660:
1659:
1653:
1645:
1637:
1631:
1630:
1610:
1604:
1603:
1567:
1561:
1560:
1550:
1540:
1516:
1510:
1505:
1495:
1472:Br. J. Pharmacol
1463:
1457:
1456:
1446:
1414:
1408:
1407:
1370:
1364:
1363:
1343:
1337:
1336:
1326:
1294:
1288:
1277:
1271:
1270:
1260:
1250:
1226:
1220:
1219:
1209:
1192:(5): 1827–1830.
1177:
1171:
1170:
1134:
1128:
1127:
1117:
1093:
1087:
1081:
1066:
1065:
1063:
1061:
1056:. 13 March 2019
1050:
857:phospholipase A2
838:second World War
757:, it is used as
755:sclerosing agent
658:
657:
598:
578:
566:
560:
557:
551:
545:
528:
517:
506:
505:
491:
489:
473:
467:
446:
426:
406:
386:
366:
346:
326:
316:
315:
301:
239:
208:
198:
177:
144:
137:
135:
131:
125:
118:
114:
111:
105:
103:
62:
38:
30:
21:
5226:
5225:
5221:
5220:
5219:
5217:
5216:
5215:
5206:Aromatic amines
5156:
5155:
5154:
5149:
5101:
5071:
5061:
5032:Diphenhydramine
5001:
4991:
4933:
4910:
4890:
4880:
4860:
4850:
4810:
4787:
4775:
4663:Normetanephrine
4629:
4619:
4579:
4569:
4509:
4499:
4436:
4426:
4396:
4379:
4368:
4366:Phenethylamines
4352:
4251:
4126:
4122:Tranylcypromine
3959:Normetanephrine
3922:
3913:
3894:
3884:
3780:
3763:
3752:
3722:
3717:
3716:
3701:Clinical trials
3676:
3657:Hexylresorcinol
3567:
3508:
3423:
3364:
3362:
3346:
3260:
3225:
3213:
3106:
3094:phosphonic acid
3079:
3073:Triclabendazole
3044:
3042:Antitrematodals
3027:
3005:
2975:
2970:
2969:
2954:Clinical trials
2929:
2894:
2874:Dientamoebiasis
2868:
2837:
2753:
2730:
2657:
2624:
2611:
2549:Trypanosomiasis
2534:
2517:
2487:
2482:
2481:
2466:Clinical trials
2445:
2428:
2417:
2400:
2385:
2359:
2337:
2331:
2281:
2271:
2220:
2187:
2176:
2159:
2136:
2098:DHFR inhibitors
2079:
2049:
2023:
1976:Aminoquinolines
1966:
1956:
1928:
1895:
1877:
1845:
1832:
1821:
1814:
1796:
1759:
1754:
1745:
1744:
1740:
1724:
1720:
1704:
1703:
1667:
1663:
1647:
1646:
1638:
1634:
1612:
1611:
1607:
1568:
1564:
1517:
1513:
1464:
1460:
1415:
1411:
1371:
1367:
1344:
1340:
1295:
1291:
1278:
1274:
1241:(39): 6366–70.
1227:
1223:
1178:
1174:
1139:Br. J. Haematol
1135:
1131:
1094:
1090:
1082:
1069:
1059:
1057:
1052:
1051:
1047:
1043:
1016:
1000:
965:Fallopian tubes
938:
892:
880:
822:
817:
785:
766:toxic psychosis
697:
653:
651:
646:
643:
638:
633:
632:
621:
618:
613:
612:
601:
576:
563:
554:
548:
509:
485:
477:
449:
429:
409:
389:
369:
349:
329:
312:
304:
284:
281:
260:
259:
237:
226:Protein binding
218:Pharmacokinetic
212:
126:
115:
109:
106:
63:
61:
51:
39:
28:
23:
22:
15:
12:
11:
5:
5224:
5214:
5213:
5208:
5203:
5198:
5193:
5188:
5183:
5178:
5173:
5168:
5151:
5150:
5110:
5107:
5106:
5103:
5102:
5100:
5099:
5090:
5089:
5076:
5074:
5063:
5062:
5060:
5059:
5054:
5049:
5044:
5039:
5034:
5029:
5020:
5019:
5006:
5004:
4993:
4992:
4990:
4989:
4984:
4979:
4974:
4969:
4964:
4955:
4954:
4938:
4936:
4922:
4916:
4915:
4912:
4911:
4909:
4908:
4895:
4893:
4882:
4881:
4879:
4878:
4865:
4863:
4852:
4851:
4849:
4848:
4843:
4838:
4829:
4828:
4815:
4813:
4799:
4781:
4780:
4777:
4776:
4774:
4773:
4768:
4763:
4758:
4753:
4748:
4743:
4738:
4729:
4728:
4719:
4710:
4701:
4692:
4683:
4674:
4665:
4659:Norepinephrine
4656:
4647:
4634:
4632:
4621:
4620:
4618:
4617:
4612:
4607:
4598:
4597:
4584:
4582:
4571:
4570:
4568:
4567:
4562:
4557:
4552:
4547:
4542:
4537:
4528:
4527:
4514:
4512:
4501:
4500:
4498:
4497:
4492:
4487:
4482:
4477:
4475:3-Iodotyrosine
4472:
4467:
4458:
4457:
4441:
4439:
4428:
4427:
4425:
4424:
4415:
4414:
4401:
4399:
4385:
4381:norepinephrine
4362:
4361:
4358:
4357:
4354:
4353:
4351:
4350:
4345:
4340:
4331:
4326:
4321:
4316:
4311:
4306:
4301:
4296:
4291:
4286:
4281:
4273:
4268:
4256:
4253:
4252:
4250:
4249:
4244:
4239:
4234:
4229:
4224:
4219:
4214:
4212:Methylene blue
4209:
4183:
4178:
4173:
4171:CX157 (Tyrima)
4168:
4163:
4158:
4153:
4148:
4143:
4131:
4128:
4127:
4125:
4124:
4119:
4114:
4109:
4104:
4099:
4094:
4089:
4084:
4079:
4074:
4069:
4064:
4059:
4054:
4049:
4044:
4039:
4034:
4029:
4024:
4019:
4014:
4009:
4004:Non-selective:
3997:
3996:
3987:
3978:
3969:
3956:
3947:
3934:
3903:
3897:
3886:
3885:
3883:
3882:
3877:
3872:
3867:
3862:
3853:
3852:
3843:
3831:
3829:Phenethylamine
3822:
3810:
3801:
3785:
3783:
3769:
3765:
3764:
3751:
3750:
3743:
3736:
3728:
3719:
3718:
3715:
3714:
3713:
3712:
3709:
3698:
3692:
3686:
3685:
3682:
3681:
3678:
3677:
3675:
3674:
3669:
3667:Tribendimidine
3664:
3659:
3654:
3649:
3648:
3647:
3635:
3634:
3633:
3625:benzylammonium
3621:
3620:
3619:
3607:
3606:
3605:
3593:
3592:
3591:
3586:
3575:
3573:
3569:
3568:
3566:
3565:
3564:
3563:
3553:
3548:
3543:
3538:
3537:
3536:
3518:
3516:
3510:
3509:
3507:
3506:
3505:
3504:
3499:
3482:
3481:
3480:
3475:
3470:
3460:
3455:
3450:
3437:
3435:
3425:
3424:
3422:
3421:
3420:
3419:
3414:
3412:Ciclobendazole
3409:
3404:
3399:
3394:
3381:
3379:
3369:
3356:
3355:
3352:
3351:
3348:
3347:
3345:
3344:
3343:
3342:
3330:
3329:
3328:
3316:
3315:
3314:
3302:
3301:
3300:
3292:salicylanilide
3288:
3287:
3286:
3268:
3266:
3262:
3261:
3259:
3258:
3257:
3256:
3243:
3241:
3231:
3219:
3218:
3215:
3214:
3212:
3211:
3210:
3209:
3204:
3191:
3190:
3189:
3184:
3172:
3171:
3170:
3158:
3157:
3156:
3144:
3143:
3142:
3137:
3127:
3125:Arpraziquantel
3114:
3112:
3108:
3107:
3105:
3104:
3103:
3102:
3089:
3087:
3085:AChE inhibitor
3081:
3080:
3078:
3077:
3076:
3075:
3062:
3060:
3050:
3035:
3029:
3028:
3008:Antiparasitics
3004:
3003:
2996:
2989:
2981:
2972:
2971:
2968:
2967:
2966:
2965:
2962:
2951:
2945:
2939:
2938:
2935:
2934:
2931:
2930:
2928:
2927:
2917:
2907:
2896:
2895:
2888:
2882:nitroimidazole
2878:
2876:
2870:
2869:
2867:
2866:
2851:nitroimidazole
2847:
2845:
2843:Trichomoniasis
2839:
2838:
2836:
2835:
2824:
2823:
2813:
2802:
2801:
2791:
2780:nitroimidazole
2776:
2774:
2765:
2759:
2758:
2755:
2754:
2752:
2751:
2748:Amphotericin B
2740:
2738:
2732:
2731:
2729:
2728:
2718:
2708:
2683:
2682:
2679:Amphotericin B
2671:
2669:
2663:
2662:
2659:
2658:
2656:
2655:
2645:
2638:nitroimidazole
2634:
2632:
2630:Chagas disease
2626:
2625:
2623:
2622:
2615:nitroimidazole
2612:
2601:
2591:
2573:
2562:
2560:
2551:
2542:
2536:
2535:
2520:Antiparasitics
2516:
2515:
2508:
2501:
2493:
2484:
2483:
2480:
2479:
2478:
2477:
2474:
2463:
2457:
2451:
2450:
2447:
2446:
2444:
2443:
2437:Blastocystosis
2433:
2431:
2423:
2422:
2419:
2418:
2416:
2415:
2405:
2403:
2395:
2394:
2391:
2390:
2387:
2386:
2384:
2383:
2377:
2375:
2369:
2368:
2365:
2364:
2361:
2360:
2358:
2357:
2354:
2351:
2348:
2345:
2341:
2339:
2333:
2332:
2330:
2329:
2324:
2319:
2313:
2307:
2301:
2295:
2293:
2283:
2277:
2276:
2273:
2272:
2270:
2269:
2264:
2259:
2254:
2249:
2244:
2239:
2228:
2226:
2222:
2221:
2219:
2218:
2213:
2208:
2203:
2198:
2192:
2190:
2182:
2181:
2178:
2177:
2175:
2174:
2167:
2165:
2164:Co-formulation
2161:
2160:
2158:
2157:
2152:
2146:
2144:
2138:
2137:
2135:
2134:
2133:
2132:
2127:
2125:chlorproguanil
2114:
2113:
2108:
2102:
2100:
2091:
2085:
2084:
2081:
2080:
2078:
2077:
2071:
2070:
2069:
2068:
2057:
2055:
2051:
2050:
2048:
2047:
2042:
2037:
2031:
2029:
2025:
2024:
2022:
2021:
2016:
2011:
2001:
2000:
1995:
1990:
1980:
1978:
1969:
1958:
1949:
1940:
1934:
1933:
1930:
1929:
1927:
1926:
1921:
1916:
1911:
1905:
1903:
1897:
1896:
1894:
1893:
1887:
1885:
1879:
1878:
1876:
1875:
1862:
1860:
1851:
1835:
1824:
1816:
1815:
1807:Chromalveolata
1799:Antiparasitics
1795:
1794:
1787:
1780:
1772:
1766:
1765:
1758:
1757:External links
1755:
1753:
1752:
1738:
1732:Indian Express
1718:
1661:
1632:
1605:
1562:
1531:(11): 2413–5.
1525:PLOS Pathogens
1511:
1458:
1429:(15): 8462–9.
1409:
1382:(12): 2413–5.
1365:
1338:
1309:(10): 4894–7.
1289:
1272:
1221:
1172:
1145:(2): 380–385.
1129:
1108:(4): 299–303.
1088:
1067:
1044:
1042:
1039:
1038:
1037:
1032:
1027:
1022:
1015:
1012:
999:
996:
953:uterine cavity
945:over its use.
937:
934:
930:in vivo effect
910:United Kingdom
891:
888:
879:
876:
862:Scientists at
821:
818:
816:
813:
807:and activates
784:
781:
777:epifluorescent
696:
693:
667:, also called
660:
659:
648:
647:
645:
644:
641:
639:
636:
628:
627:
626:
623:
622:
620:
619:
616:
608:
607:
606:
603:
602:
600:
599:
591:
589:
581:
580:
574:
568:
567:
561:
552:
546:
541:
535:
534:
530:
529:
519:
511:
510:
508:
507:
494:
492:
479:
478:
476:
475:
459:
457:
451:
450:
448:
447:
439:
437:
431:
430:
428:
427:
419:
417:
411:
410:
408:
407:
399:
397:
391:
390:
388:
387:
379:
377:
371:
370:
368:
367:
359:
357:
351:
350:
348:
347:
339:
337:
331:
330:
328:
327:
319:
317:
306:
305:
303:
302:
294:
292:
286:
285:
283:
282:
263:
255:
254:
253:
250:
249:
245:
244:
241:
232:
231:
228:
222:
221:
214:
213:
211:
210:
187:
185:
179:
178:
171:
161:
160:
157:
151:
150:
146:
145:
128:
127:
42:
40:
33:
26:
9:
6:
4:
3:
2:
5223:
5212:
5209:
5207:
5204:
5202:
5201:Phenol ethers
5199:
5197:
5194:
5192:
5189:
5187:
5184:
5182:
5179:
5177:
5174:
5172:
5169:
5167:
5164:
5163:
5161:
5147:
5146:
5142:
5138:
5134:
5133:Serotonergics
5130:
5129:Melatonergics
5126:
5125:Dopaminergics
5122:
5118:
5115:
5108:
5098:
5095:
5092:
5091:
5088:
5084:
5081:
5078:
5077:
5075:
5070:
5064:
5058:
5055:
5053:
5050:
5048:
5045:
5043:
5040:
5038:
5035:
5033:
5030:
5028:
5025:
5022:
5021:
5018:
5014:
5011:
5008:
5007:
5005:
5000:
4994:
4988:
4985:
4983:
4980:
4978:
4975:
4973:
4970:
4968:
4965:
4963:
4960:
4957:
4956:
4953:
4949:
4943:
4940:
4939:
4937:
4932:
4926:
4923:
4921:
4917:
4907:
4903:
4900:
4897:
4896:
4894:
4889:
4883:
4877:
4873:
4870:
4867:
4866:
4864:
4859:
4853:
4847:
4844:
4842:
4839:
4837:
4834:
4831:
4830:
4827:
4823:
4820:
4817:
4816:
4814:
4809:
4803:
4800:
4796:
4792:
4786:
4782:
4772:
4769:
4767:
4764:
4762:
4759:
4757:
4754:
4752:
4749:
4747:
4744:
4742:
4739:
4737:
4734:
4731:
4730:
4727:
4723:
4720:
4718:
4714:
4711:
4709:
4705:
4702:
4700:
4696:
4693:
4691:
4687:
4684:
4682:
4678:
4675:
4673:
4669:
4666:
4664:
4660:
4657:
4655:
4651:
4648:
4646:
4642:
4639:
4636:
4635:
4633:
4628:
4622:
4616:
4613:
4611:
4608:
4606:
4603:
4600:
4599:
4596:
4592:
4589:
4586:
4585:
4583:
4578:
4572:
4566:
4563:
4561:
4558:
4556:
4553:
4551:
4548:
4546:
4543:
4541:
4538:
4536:
4533:
4530:
4529:
4526:
4522:
4519:
4516:
4515:
4513:
4508:
4502:
4496:
4493:
4491:
4488:
4486:
4483:
4481:
4478:
4476:
4473:
4471:
4468:
4466:
4463:
4460:
4459:
4456:
4449:
4446:
4443:
4442:
4440:
4435:
4429:
4423:
4420:
4417:
4416:
4413:
4409:
4408:Phenylalanine
4406:
4403:
4402:
4400:
4395:
4389:
4386:
4382:
4377:
4373:
4367:
4363:
4349:
4346:
4344:
4341:
4339:
4332:
4330:
4327:
4325:
4322:
4320:
4317:
4315:
4312:
4310:
4307:
4305:
4302:
4300:
4297:
4295:
4292:
4290:
4287:
4285:
4282:
4280:
4274:
4272:
4269:
4267:
4264:
4261:
4258:
4257:
4254:
4248:
4245:
4243:
4240:
4238:
4235:
4233:
4230:
4228:
4225:
4223:
4220:
4218:
4215:
4213:
4210:
4207:
4203:
4199:
4195:
4191:
4187:
4184:
4182:
4179:
4177:
4174:
4172:
4169:
4167:
4164:
4162:
4159:
4157:
4154:
4152:
4149:
4147:
4144:
4142:
4139:
4136:
4133:
4132:
4129:
4123:
4120:
4118:
4115:
4113:
4110:
4108:
4105:
4103:
4100:
4098:
4095:
4093:
4090:
4088:
4085:
4083:
4080:
4078:
4075:
4073:
4072:Metfendrazine
4070:
4068:
4065:
4063:
4060:
4058:
4055:
4053:
4052:Isocarboxazid
4050:
4048:
4045:
4043:
4040:
4038:
4035:
4033:
4030:
4028:
4025:
4023:
4020:
4018:
4017:Echinopsidine
4015:
4013:
4010:
4008:
4005:
4002:
3999:
3998:
3995:
3991:
3988:
3986:
3982:
3979:
3977:
3973:
3970:
3968:
3964:
3960:
3957:
3955:
3951:
3948:
3946:
3942:
3938:
3935:
3933:
3929:
3926:
3921:
3912:
3905:
3904:
3901:
3898:
3893:
3887:
3881:
3878:
3876:
3873:
3871:
3868:
3866:
3863:
3861:
3858:
3855:
3854:
3851:
3847:
3844:
3842:
3838:
3832:
3830:
3826:
3825:Phenylalanine
3823:
3821:
3817:
3811:
3809:
3805:
3802:
3800:
3796:
3790:
3787:
3786:
3784:
3779:
3773:
3770:
3766:
3762:
3759:
3756:
3749:
3744:
3742:
3737:
3735:
3730:
3729:
3726:
3710:
3708:
3705:
3704:
3702:
3699:
3696:
3693:
3691:
3688:
3687:
3683:
3673:
3670:
3668:
3665:
3663:
3660:
3658:
3655:
3653:
3650:
3646:
3643:
3642:
3641:
3640:
3636:
3632:
3629:
3628:
3627:
3626:
3622:
3618:
3615:
3614:
3613:
3612:
3608:
3604:
3601:
3600:
3599:
3598:
3594:
3590:
3587:
3585:
3582:
3581:
3580:
3577:
3576:
3574:
3572:Other/unknown
3570:
3561:
3557:
3554:
3552:
3549:
3547:
3544:
3542:
3539:
3535:
3532:
3531:
3530:
3527:
3526:
3525:
3524:
3520:
3519:
3517:
3515:
3511:
3503:
3500:
3497:
3493:
3490:
3489:
3488:
3487:
3483:
3479:
3476:
3474:
3471:
3468:
3464:
3461:
3459:
3456:
3454:
3451:
3449:
3446:
3445:
3444:
3443:
3439:
3438:
3436:
3434:
3433:GABA receptor
3430:
3426:
3418:
3415:
3413:
3410:
3408:
3405:
3403:
3400:
3398:
3395:
3393:
3390:
3389:
3388:
3387:
3386:benzimidazole
3383:
3382:
3380:
3378:
3373:
3370:
3367:
3361:
3357:
3341:
3338:
3337:
3336:
3335:
3331:
3327:
3324:
3323:
3322:
3321:
3320:butyrophenone
3317:
3313:
3310:
3309:
3308:
3307:
3306:aminoacridine
3303:
3299:
3296:
3295:
3294:
3293:
3289:
3284:
3280:
3277:
3276:
3275:
3274:
3270:
3269:
3267:
3265:Other/unknown
3263:
3255:
3252:
3251:
3250:
3249:
3248:benzimidazole
3245:
3244:
3242:
3240:
3235:
3232:
3229:
3224:
3223:Anticestodals
3220:
3208:
3207:Tartar emetic
3205:
3203:
3200:
3199:
3198:
3196:
3192:
3188:
3185:
3183:
3180:
3179:
3178:
3177:
3173:
3169:
3166:
3165:
3164:
3163:
3159:
3155:
3152:
3151:
3150:
3149:
3145:
3141:
3138:
3135:
3131:
3128:
3126:
3123:
3122:
3121:
3120:
3116:
3115:
3113:
3111:Other/unknown
3109:
3101:
3098:
3097:
3096:
3095:
3091:
3090:
3088:
3086:
3082:
3074:
3071:
3070:
3069:
3068:
3067:benzimidazole
3064:
3063:
3061:
3059:
3054:
3051:
3048:
3043:
3039:
3036:
3034:
3030:
3025:
3021:
3017:
3013:
3012:Anthelmintics
3009:
3002:
2997:
2995:
2990:
2988:
2983:
2982:
2979:
2963:
2961:
2958:
2957:
2955:
2952:
2949:
2946:
2944:
2941:
2940:
2936:
2925:
2921:
2918:
2915:
2911:
2908:
2905:
2901:
2898:
2897:
2892:
2889:
2887:
2886:Metronidazole
2883:
2880:
2879:
2877:
2875:
2871:
2864:
2860:
2859:Metronidazole
2856:
2852:
2849:
2848:
2846:
2844:
2840:
2833:
2829:
2828:aminoacridine
2826:
2825:
2821:
2817:
2814:
2811:
2807:
2804:
2803:
2799:
2795:
2794:benzimidazole
2792:
2789:
2785:
2784:Metronidazole
2781:
2778:
2777:
2775:
2773:
2769:
2766:
2764:
2760:
2749:
2745:
2742:
2741:
2739:
2737:
2733:
2726:
2722:
2719:
2716:
2712:
2709:
2706:
2702:
2699:
2698:
2697:
2695:
2691:
2687:
2680:
2676:
2673:
2672:
2670:
2668:
2667:Leishmaniasis
2664:
2653:
2649:
2646:
2643:
2639:
2636:
2635:
2633:
2631:
2627:
2620:
2616:
2613:
2609:
2605:
2602:
2599:
2595:
2592:
2589:
2585:
2581:
2577:
2574:
2571:
2567:
2564:
2563:
2561:
2559:
2555:
2552:
2550:
2546:
2543:
2541:
2540:Discicristata
2537:
2532:
2528:
2525:
2521:
2514:
2509:
2507:
2502:
2500:
2495:
2494:
2491:
2475:
2473:
2470:
2469:
2467:
2464:
2461:
2458:
2456:
2453:
2452:
2448:
2442:
2441:metronidazole
2438:
2435:
2434:
2432:
2430:
2424:
2414:
2410:
2409:Balantidiasis
2407:
2406:
2404:
2402:
2396:
2382:
2379:
2378:
2376:
2374:
2370:
2355:
2352:
2349:
2347:artesunate/SP
2346:
2343:
2342:
2340:
2334:
2328:
2325:
2323:
2320:
2317:
2314:
2311:
2308:
2305:
2302:
2300:
2297:
2296:
2294:
2292:
2287:
2284:
2278:
2268:
2265:
2263:
2260:
2258:
2255:
2253:
2250:
2248:
2245:
2243:
2240:
2237:
2233:
2230:
2229:
2227:
2223:
2217:
2214:
2212:
2209:
2207:
2204:
2202:
2199:
2197:
2194:
2193:
2191:
2189:
2186:Sesquiterpene
2183:
2172:
2169:
2168:
2166:
2162:
2156:
2153:
2151:
2148:
2147:
2145:
2143:
2139:
2131:
2128:
2126:
2123:
2122:
2121:
2120:
2116:
2115:
2112:
2109:
2107:
2106:pyrimethamine
2104:
2103:
2101:
2099:
2095:
2092:
2090:
2086:
2076:
2073:
2072:
2067:
2064:
2063:
2062:
2059:
2058:
2056:
2052:
2046:
2043:
2041:
2038:
2036:
2033:
2032:
2030:
2026:
2020:
2017:
2015:
2012:
2010:
2006:
2003:
2002:
1999:
1996:
1994:
1991:
1989:
1985:
1982:
1981:
1979:
1977:
1973:
1970:
1968:
1962:
1959:
1953:
1950:
1948:
1944:
1941:
1939:
1935:
1925:
1922:
1920:
1917:
1915:
1912:
1910:
1909:pyrimethamine
1907:
1906:
1904:
1902:
1901:Toxoplasmosis
1898:
1892:
1889:
1888:
1886:
1884:
1880:
1873:
1869:
1868:
1864:
1863:
1861:
1859:
1855:
1852:
1849:
1848:Coccidiostats
1843:
1839:
1836:
1834:
1828:
1825:
1823:
1817:
1812:
1808:
1804:
1800:
1793:
1788:
1786:
1781:
1779:
1774:
1773:
1770:
1764:
1761:
1760:
1749:. 2019-01-26.
1748:
1742:
1733:
1729:
1722:
1714:
1708:
1700:
1696:
1692:
1688:
1684:
1680:
1677:(2): 139–44.
1676:
1672:
1665:
1657:
1651:
1643:
1636:
1628:
1624:
1620:
1616:
1609:
1601:
1597:
1593:
1589:
1585:
1581:
1578:(4): 275–90.
1577:
1573:
1566:
1558:
1554:
1549:
1544:
1539:
1534:
1530:
1526:
1522:
1515:
1509:
1503:
1499:
1494:
1489:
1485:
1481:
1478:(3): 386–93.
1477:
1473:
1469:
1462:
1454:
1450:
1445:
1440:
1436:
1432:
1428:
1424:
1420:
1413:
1405:
1401:
1397:
1393:
1389:
1385:
1381:
1377:
1369:
1361:
1357:
1353:
1349:
1342:
1334:
1330:
1325:
1320:
1316:
1312:
1308:
1304:
1300:
1293:
1287:
1286:
1281:
1276:
1268:
1264:
1259:
1254:
1249:
1244:
1240:
1236:
1232:
1225:
1217:
1213:
1208:
1203:
1199:
1195:
1191:
1187:
1183:
1176:
1168:
1164:
1160:
1156:
1152:
1148:
1144:
1140:
1133:
1125:
1121:
1116:
1111:
1107:
1103:
1099:
1092:
1085:
1080:
1078:
1076:
1074:
1072:
1055:
1049:
1045:
1036:
1033:
1031:
1028:
1026:
1023:
1021:
1018:
1017:
1011:
1009:
1005:
995:
993:
989:
985:
980:
978:
972:
970:
966:
962:
958:
954:
950:
946:
943:
942:sterilization
933:
931:
927:
923:
919:
915:
914:United States
911:
907:
903:
902:
897:
887:
885:
878:Anthelmintics
875:
873:
869:
865:
860:
858:
854:
850:
846:
845:antiprotozoal
841:
839:
835:
826:
820:Antiprotozoal
812:
810:
806:
802:
800:
794:
790:
780:
778:
773:
771:
767:
762:
760:
756:
751:
750:
746:
742:
737:
735:
734:metronidazole
730:
728:
724:
723:antirheumatic
720:
719:antiprotozoal
713:
709:
705:
701:
692:
690:
686:
682:
678:
674:
670:
666:
656:
649:
640:
635:
634:
631:
624:
615:
614:
611:
604:
597:
593:
592:
590:
587:
582:
575:
573:
569:
542:
540:
536:
531:
527:
523:
520:
518:
516:ECHA InfoCard
512:
504:
500:
499:DTXSID7022627
496:
495:
493:
484:
480:
472:
471:RCSB PDB
466:
461:
460:
458:
456:
452:
445:
441:
440:
438:
436:
432:
425:
421:
420:
418:
416:
412:
405:
401:
400:
398:
396:
392:
385:
381:
380:
378:
376:
372:
365:
361:
360:
358:
356:
352:
345:
341:
340:
338:
336:
332:
325:
321:
320:
318:
311:
307:
300:
296:
295:
293:
291:
287:
279:
275:
271:
267:
262:
261:
258:
251:
246:
242:
240:
233:
229:
227:
223:
219:
215:
207:
202:
197:
192:
189:
188:
186:
184:
180:
176:
172:
170:
166:
162:
158:
156:
152:
149:Clinical data
147:
143:
138:
124:
121:
113:
102:
99:
95:
92:
88:
85:
81:
78:
74:
71: –
70:
66:
65:Find sources:
59:
55:
49:
48:
43:This article
41:
37:
32:
31:
19:
5196:Chloroarenes
5113:
5112:
5093:
5079:
5023:
5009:
4987:Tritoqualine
4958:
4941:
4898:
4868:
4832:
4818:
4766:Quinalizarin
4751:Neluxicapone
4732:
4672:Metanephrine
4637:
4601:
4587:
4550:Fusaric acid
4531:
4517:
4485:Bulbocapnine
4461:
4444:
4418:
4404:
4348:Tisolagiline
4343:Sembragiline
4334:Selegiline (
4262:
4259:
4237:Sercloremine
4217:Metralindole
4137:
4134:
4112:Procarbazine
4107:Pivhydrazine
4097:Pheniprazine
4022:Furazolidone
4003:
4000:
3937:Metanephrine
3906:
3856:
3788:
3768:Non-specific
3637:
3623:
3609:
3595:
3578:
3521:
3484:
3463:Eprinomectin
3440:
3417:Flubendazole
3407:Fenbendazole
3402:Tiabendazole
3384:
3340:Dichlorophen
3334:chlorophenol
3332:
3318:
3304:
3290:
3279:Praziquantel
3271:
3246:
3193:
3176:thioxanthone
3174:
3160:
3146:
3130:Praziquantel
3117:
3092:
3065:
3020:endectocides
2910:tetracycline
2900:oxyquinoline
2820:Furazolidone
2810:Nitazoxanide
2684:
2642:Benznidazole
2619:Fexinidazole
2588:Tryparsamide
2570:Eflornithine
2522:directed at
2413:tetracycline
2306:/piperaquine
2262:pyronaridine
2256:
2242:tetracycline
2142:Sulfonamides
2117:
2075:halofantrine
2066:+ artemether
2061:lumefantrine
1938:Aconoidasida
1914:sulfadiazine
1883:Isosporiasis
1872:nitazoxanide
1865:
1741:
1731:
1721:
1707:cite journal
1674:
1670:
1664:
1650:cite journal
1641:
1635:
1618:
1614:
1608:
1575:
1571:
1565:
1528:
1524:
1514:
1475:
1471:
1461:
1426:
1422:
1412:
1379:
1375:
1368:
1354:(7): 403–8.
1351:
1347:
1341:
1306:
1302:
1292:
1283:
1280:"quinacrine"
1275:
1238:
1234:
1224:
1189:
1185:
1175:
1142:
1138:
1132:
1105:
1101:
1091:
1058:. Retrieved
1048:
1001:
981:
973:
947:
939:
929:
899:
893:
886:infections.
881:
861:
842:
831:
798:
786:
774:
763:
759:pneumothorax
752:
738:
731:
716:
703:
695:Medical uses
676:
672:
668:
664:
663:
652:
277:
273:
269:
265:
236:Elimination
116:
107:
97:
90:
83:
76:
64:
52:Please help
47:verification
44:
5121:Adrenergics
5094:Inhibitors:
5027:Amodiaquine
5024:Inhibitors:
4959:Inhibitors:
4833:Inhibitors:
4785:Tryptamines
4733:Inhibitors:
4668:Epinephrine
4602:Inhibitors:
4532:Inhibitors:
4480:Aquayamycin
4462:Inhibitors:
4419:Inhibitors:
4376:epinephrine
4266:Adarigiline
4260:Inhibitors:
4227:Moclobemide
4156:Brofaromine
4151:Befloxatone
4146:Bazinaprine
4135:Inhibitors:
4042:Iproclozide
4032:Hydralazine
4001:Inhibitors:
3923:Tooltip ALR
3860:Benserazide
3857:Inhibitors:
3697:from market
3611:quinolinium
3496:+fluralaner
3486:milbemycins
3442:avermectins
3397:Albendazole
3392:Mebendazole
3298:Niclosamide
3254:Albendazole
3228:taeniacides
3140:Oxamniquine
3100:Metrifonate
2950:from market
2924:Paromomycin
2914:Doxycycline
2891:Secnidazole
2855:Carnidazole
2798:Albendazole
2725:Paromomycin
2715:Miltefosine
2705:Pentamidine
2701:benzamidine
2598:Pentamidine
2594:benzamidine
2584:Melarsoprol
2462:from market
2381:clindamycin
2267:piperaquine
2252:clindamycin
2247:doxycycline
2236:+ proguanil
2201:artemisinin
2150:sulfadoxine
2111:cycloguanil
2089:Antifolates
2019:tafenoquine
1993:chloroquine
1988:amodiaquine
1955:Individual
1919:clindamycin
1867:thiazolides
1842:Conoidasida
1025:Amodiaquine
1020:Chloroquine
1006:, American
1002:During the
969:scar tissue
872:chloroquine
681:chloroquine
579: g·mol
522:100.001.371
248:Identifiers
155:Trade names
110:August 2024
69:"Mepacrine"
5160:Categories
5047:Quinacrine
4982:Naringenin
4977:Meciadanol
4948:-Histidine
4822:Tryptophan
4756:Nitecapone
4746:Entacapone
4605:CGS-19281A
4555:Nepicastat
4540:Disulfiram
4535:Bupicomide
4490:Metirosine
4338:-Deprenyl)
4329:Safinamide
4324:Rasagiline
4309:Mofegiline
4304:Milacemide
4299:Lazabemide
4294:Ladostigil
4271:Almoxatone
4247:Toloxatone
4242:Tetrindole
4232:Pirlindole
4176:Eprobemide
4166:Clorgiline
4161:Cimoxatone
4141:Amiflamine
4092:Phenelzine
4087:Paraxazone
4067:Mebanazine
4047:Iproniazid
4037:Indantadol
4027:Guineesine
4012:Caroxazone
3880:Methyldopa
3850:Tryptamine
3846:Tryptophan
3816:-Histidine
3761:modulators
3758:metabolism
3652:Ascaridole
3603:Levamisole
3584:Piperazine
3579:piperazine
3492:Moxidectin
3478:Selamectin
3473:Ivermectin
3453:Doramectin
3363:(including
3326:Desaspidin
3312:Quinacrine
3187:Lucanthone
3182:Hycanthone
3168:Niridazole
2904:Iodoquinol
2863:Tinidazole
2832:Quinacrine
2816:nitrofuran
2806:thiazolide
2788:Tinidazole
2772:Giardiasis
2652:Nifurtimox
2648:nitrofuran
2373:Babesiosis
2304:arterolane
2232:atovaquone
2211:artesunate
2196:artemether
2119:biguanides
2035:mefloquine
2009:primaquine
1967:inhibitors
1924:atovaquone
1041:References
1035:Mefloquine
961:sclerosing
849:giardiasis
797:histamine
770:mefloquine
727:sclerosing
685:mefloquine
669:quinacrine
584:3D model (
572:Molar mass
455:PDB ligand
444:ChEMBL7568
424:CHEBI:8711
384:H0C805XYDE
355:ChemSpider
290:CAS Number
257:IUPAC name
80:newspapers
27:Medication
18:Quinacrine
5191:Acridines
5114:See also:
5083:Histamine
5052:SKF-91488
5042:Metoprine
5037:Harmaline
5013:Histamine
4952:Histamine
4920:Histamine
4906:Melatonin
4872:Serotonin
4795:melatonin
4791:serotonin
4771:Tolcapone
4761:Opicapone
4610:SKF-64139
4565:Tropolone
4319:Pargyline
4279:-Deprenyl
4222:Minaprine
4202:norharman
4194:harmaline
4117:Safrazine
4082:Octamoxin
4077:Nialamide
4062:Linezolid
4057:Isoniazid
3990:Serotonin
3875:Genistein
3865:Carbidopa
3837:-Tyrosine
3820:Histamine
3808:Serotonin
3755:Monoamine
3707:Phase III
3695:Withdrawn
3631:Bephenium
3617:Pyrvinium
3560:felsantel
3551:Carbantel
3458:Emamectin
3448:Abamectin
3273:quinoline
3202:Stibophen
3197:compounds
3154:Bithionol
3119:quinoline
2960:Phase III
2948:Withdrawn
2920:neomycin
2763:Trichozoa
2576:arsenical
2566:ornithine
2527:parasites
2472:Phase III
2460:Withdrawn
2257:mepacrine
2206:artemotil
2155:sulfalene
2130:proguanil
2045:quinidine
2014:pamaquine
1376:Neurology
1060:24 August
1030:Pamaquine
977:off-label
793:protozoan
783:Mechanism
665:Mepacrine
243:5–14 days
238:half-life
169:Drugs.com
134:Mepacrine
4962:Catechin
4836:AGN-2979
4641:Dopamine
4615:SKF-7698
4545:Dopastin
4521:Dopamine
4495:Oudenone
4448:Tyrosine
4412:Tyrosine
4372:dopamine
4314:Nicotine
4181:Esuprone
4007:Benmoxin
3972:Dopamine
3841:Tyramine
3799:Dopamine
3662:Santonin
3597:thiazole
3556:Febantel
3546:Morantel
3529:Pyrantel
3195:antimony
3162:thiazole
3010: –
2721:neomycin
2524:excavata
2427:Stramen-
2188:lactones
1965:Hemozoin
1699:15179539
1627:14763179
1600:41946631
1557:19956709
1508:Abstract
1502:15655516
1453:12857915
1423:J. Virol
1404:37534686
1396:15623716
1360:14582366
1333:10775631
1267:17072963
1216:21383088
1167:24132625
1124:16623930
1014:See also
998:Skin dye
912:and the
901:in vitro
884:tapeworm
789:protozoa
673:Atabrine
655:(verify)
335:DrugBank
201:QP51AX04
183:ATC code
5057:Tacrine
4289:Ethanol
4190:harmine
4188:(e.g.,
3645:Suramin
3541:Oxantel
3377:tubulin
3239:tubulin
3058:tubulin
2744:polyene
2675:polyene
2608:Suramin
2282:nations
2040:quinine
1947:Malaria
1831:Apicom-
1691:6136433
1644:: 25–7.
1592:6109672
1548:2777304
1493:1576015
1303:J Virol
1258:4088148
1207:3088196
1159:7873389
949:Pellets
918:scrapie
868:quinine
815:History
745:discoid
729:agent.
706:(as an
677:Atebrin
539:Formula
344:DB01103
310:PubChem
299:83-89-6
203: (
199:)
193: (
191:P01AX05
94:scholar
4198:harman
3994:5-HIAA
3690:WHO-EM
3375:Binds
3237:Binds
3148:phenol
3056:Binds
3018:) and
2943:WHO-EM
2580:Atoxyl
2455:WHO-EM
2399:Cilio-
2318:(ASMQ)
2312:(ASAQ)
2280:Combi-
1957:agents
1820:Alveo-
1697:
1689:
1625:
1598:
1590:
1555:
1545:
1500:
1490:
1451:
1444:165262
1441:
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1394:
1358:
1331:
1324:112015
1321:
1265:
1255:
1214:
1204:
1165:
1157:
1122:
988:cancer
753:As an
610:SMILES
577:399.96
435:ChEMBL
404:D08179
230:80–90%
96:
89:
82:
75:
67:
4857:AANAT
4826:5-HTP
4681:MOPEG
4677:DOPEG
4650:DOPAC
3976:DOPAC
3804:5-HTP
3558:(aka
2429:opile
2401:phora
2225:Other
2054:Other
1833:plexa
1695:S2CID
1596:S2CID
1400:S2CID
1163:S2CID
926:sheep
896:prion
864:Bayer
843:This
805:NF-κB
630:InChI
586:JSmol
462:QUN (
415:ChEBI
101:JSTOR
87:books
4998:HNMT
4887:ASMT
4686:DOMA
4626:COMT
4576:PNMT
3963:MHPG
3954:DHMA
3941:MHPG
3932:DHMA
3910:ALDH
3870:DFMD
3777:AAAD
3514:NMDA
3024:QP54
2291:ACTs
2173:(SP)
2005:(8-)
1984:(4-)
1822:late
1713:link
1687:PMID
1656:link
1623:PMID
1588:PMID
1553:PMID
1498:PMID
1449:PMID
1392:PMID
1356:PMID
1329:PMID
1263:PMID
1212:PMID
1155:PMID
1120:PMID
1062:2020
957:IUCD
924:and
922:mice
851:(an
683:and
465:PDBe
395:KEGG
375:UNII
220:data
165:AHFS
73:news
5068:DAO
4930:HDC
4807:TPH
4690:VMA
4506:DBH
4393:PAH
3985:HVA
3967:VMA
3945:VMA
3919:ALR
3891:MAO
3016:P02
2736:PAM
2531:P01
1811:P01
1679:doi
1580:doi
1543:PMC
1533:doi
1488:PMC
1480:doi
1476:144
1439:PMC
1431:doi
1384:doi
1319:PMC
1311:doi
1282:at
1253:PMC
1243:doi
1202:PMC
1194:doi
1147:doi
1110:doi
990:or
920:in
809:p53
675:or
488:EPA
364:232
324:237
314:CID
206:WHO
196:WHO
56:by
5162::
5143:•
5139:•
5135:•
5131:•
5127:•
5123:•
5119:•
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